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Amelubant
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Amelubant图片
CAS NO:346735-24-8
包装与价格:
包装价格(元)
100 mg电议
500 mg电议

产品名称
BIIL 284
产品介绍

产品描述

Amelubant (BIIL 284) is a prodrug of active metabolites BIIL 260 and BIIL 315. Anti-inflammatory activity[1]. Amelubant (BIIL 284) is a potent, oral and long acting LTB4 receptor antagonist, negligibly binds to LTB4 receptor, with Kis of 221 nM and 230 nM in vital cells and membranes.

体外活性

Amelubant is a prodrug of active metabolites BIIL 260 and BIIL 315. Which are reversible and competitive LTB4 receptor antagonists, with Kis of 1.4, 1.1 nM and 1.7, 1.9 nM in vital cells and membranes, respectively[1].

Cas No.

346735-24-8

分子式

C33H34N2O5

分子量

538.63

别名

BIIL 284

储存和溶解度

(< 1 mg/ml refers to the product slightly soluble or insoluble )
Powder: -20°C for 3 years
In solvent: -80°C for 2 years