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Acrivastine
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Acrivastine图片
CAS NO:87848-99-5
包装与价格:
包装价格(元)
5 mg电议
10 mg电议
25 mg电议
50 mg电议
100 mg电议
1 mL*10 mM(in DMSO)电议

产品名称
Semprex
Acrivastin
BW825C
阿伐斯汀
产品介绍
Acrivastine 是一种短效组胺 1 受体拮抗剂,可用于研究过敏性鼻炎。

产品描述

Acrivastine is a short-acting histamine 1 receptor antagonist.

体内活性

Acrivastine (usually 8mg three times daily) is an effective and well-tolerated antihistamine in the treatment of chronic urticaria and allergic rhinitis. Acrivastine causes less drowsiness than clemastine, the incidence of adverse effects being indistinguishable from that with placebo or terfenadine. In the treatment of dermatoses in which histamine has a pathogenetic role, the efficacy of acrivastine is superior to that of placebo and similar to that of usual dosages of clemastine, hydroxyzine, chlorpheniramine, cyproheptadine or terfenadine [1]. Both 4 mg and 8 mg acrivastine alleviate the symptoms of seasonal allergic rhinitis with significant improvements in the symptom scores for sneezing, running nose and the calculated overall score. In addition, 8 mg acrivastine reduces the symptom scores for watery eyes and itchy throat. Acrivastine is both well tolerated and effective in the treatment of seasonal allergic rhinitis [2].

Cas No.

87848-99-5

分子式

C22H24N2O2

分子量

348.446

别名

Semprex;Acrivastin;BW825C;阿伐斯汀

储存和溶解度

DMSO:10 mg/mL,warmed&ultrasonic
Powder: -20°C for 3 years
In solvent: -80°C for 2 years