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APNEA
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
APNEA图片
CAS NO:89705-21-5
包装与价格:
包装价格(元)
5 mg电议
1 mL*10 mM(in DMSO)电议

产品名称
N6-[2-(4-氨基苯基)乙基]腺嘌呤
(2R,3R,4S,5R)-2-[6-[2-(4-aminophenyl)ethylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol
产品介绍
APNEA 是腺苷 A3 受体的非选择性激动剂。

产品描述

APNEA is a non-selective agonist of adenosine A3 receptor.

体外活性

APNEA at the subprotective dose of 1 mg/kg against electroconvulsions, significantly potentiated the anticonvulsive action of phenobarbital, diphenylhydantoin and valproate against maximal electroshock, being ineffective at lower doses[2].

体内活性

APNEA (0.0039-1 mg/kg) enhanced the protective activity of carbamazepine. APNEA (0.0156 and 1 mg/kg) administered alone or in combination with carbamazepine significantly decreased the body temperature and impaired long-term memory[2].

Cas No.

89705-21-5

分子式

C18H22N6O4

分子量

386.41

别名

N6-[2-(4-氨基苯基)乙基]腺嘌呤;(2R,3R,4S,5R)-2-[6-[2-(4-aminophenyl)ethylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol

储存和溶解度

DMSO:200 mg/mL (517.58 mM),Need ultrasonic
Powder: -20°C for 3 years
In solvent: -80°C for 2 years