PBRM1-BD2-IN-7 是一种选择性和细胞活性的 PBRM1 溴化域抑制剂。PBRM1-BD2-IN-7 对 PBRM1-BD2 具有抑制活性，IC50 值为 0.29 μM。PBRM1-BD2-IN-7 可用于癌症的研究。

PBRM1-BD2-IN-7 is a selective and cell-active polybromo-1 (PBRM1) bromodomain inhibitor. PBRM1-BD2-IN-7 has inhibitory activity for PBRM1-BD2 with an IC50 value of 0.29 μM. PBRM1-BD2-IN-7 can be used for the research of cancer.

PBRM1-BD2-IN-7 (0, 0.1, 1, and 10 μM; 5 days) selectively inhibit growth of a PBRM1-dependent prostate cancer cell line. PBRM1-BD2-IN-7 has inhibitory activity for PBRM1-BD2 with IC50 value of 0.29 μM[1].

2819989-68-7

C16H15ClN2O

286.76

(< 1 mg/ml refers to the product slightly soluble or insoluble )
Powder: -20°C for 3 years
In solvent: -80°C for 2 years