Mulberrin 能够抑制有机阴离子转运多肽 2B1 介导的雌酮-3-硫酸盐摄取(IC50:1.8±1.5 μM)。
产品描述
Mulberrin is an inhibitor of OATP2B1-mediated estrone-3-sulfate (E3S) uptake (IC50: 1.8 ±1.5 μM).
体外活性
Mulberrin is a strong inhibitor of OATP2B1 with more than 80% inhibition. Mulberrin also inhibits organic anion-transporting polypeptide (OATP)-mediated uptake of Fluvastatin, Atorvastatin, and Rosuvastatin.
Cas No.
62949-79-5
分子式
C25H26O6
分子量
422.47
别名
桑黄酮;Kuwanon C
储存和溶解度
DMSO:Soluble
Powder: -20°C for 3 years
In solvent: -80°C for 2 years