CetRORelix diacetate 是GnRH受体的强效拮抗剂(IC50:1.21 nM)。

Cetrorelix diacetate is is a gonadotropin-releasing hormone antagonist. It works by blocking the action of GnRH upon the pituitary, thus rapidly suppressing the production and action of luteinizing hormone (LH) and follicle-stimulating hormone (FSH).

130143-01-0

C72H96ClN17O16

1491.09

醋酸西曲瑞克;SB-075 acetate;NS-75A;SB-075 diacetate;Cetrorelix acetate;NS-75A diacetate

H2O:2 mg/mL (1.34 mM),Need ultrasonic
DMSO:50 mg/mL (33.53 mM),Need ultrasonic
Powder: -20°C for 3 years
In solvent: -80°C for 2 years