OMDM-5 是有效的、选择性的anandamide 细胞摄取抑制剂，Ki为 4.8 μM。它是VR1 (TRPV1)激动剂，EC50为 75 nM，显示出对大麻素 1 型受体 (CB1) 的弱配体活性 (Ki=4.9 μM)。

OMDM-5 is a potent vanilloid receptor type 1 (TRPV1, EC50 = 75 nM) agonist, showing weak ligand activity at cannabinoid type 1 receptor (CB1, Ki=4.9 μM). OMDM-5 is a selective anandamide cellular uptake (ACU) inhibitor(Ki = 4.8 μM).

616884-66-3

C26H44N2O3

432.64

DMSO:65 mg/ml (150.24 mM)
Powder: -20°C for 3 years
In solvent: -80°C for 2 years