LPA2 antagonist 2 (H2L 5226501) is a specific LPA2 antagonist with an IC50 of 28.3 nM and a Ki of 21.1 nM. LPA2 antagonist 2 is ＞480-fold more specific than LPA3 (IC50 of 13.85 μM). References: [1]. Fells JI, et al. Identification of non-lipid LPA3 antagonists by virtual screening. Bioorg Med Chem. 2008 Jun 1;16(11):6207-17.

纯度：≥98%

CAS：36840-10-5