S26131 是一种选择性的褪黑激素配体 MT1 和 MT2 拮抗剂,对 MT1 和 MT2 的Ki值分别为 0.5 和 112 nM。
产品描述
S26131 behaves as an antagonist on MT1 and MT2 receptors with Ki of 0.5 and 112 nM respectively.
体外活性
S26131 is an effective and selective antagonist of MT1 and MT2 with KBs of 5.32 and 143 nM, respectively[1].
Cas No.
296280-56-3
分子式
C31H34N2O4
分子量
498.61
别名
N-[2-[7-[3-[8-(2-acetamidoethyl)naphthalen-2-yl]oxypropoxy]naphthalen-1-yl]ethyl]acetamide
储存和溶解度
DMSO:25 mg/mL (50.14 mM),Need ultrasonic
Powder: -20°C for 3 years
In solvent: -80°C for 2 years