Bremelanotide Acetate 是 α-MSH 的合成肽类似物，是黑素皮质素受体 MC3R 和 MC4R 的激动剂，有用于性功能障碍的研究潜力。

Bremelanotide is an agonist of melanocortin receptor (MCR) .

Treatment with Bremelanotide?(100 or 200 μg/kg) significantly increased proceptive solicitations in females primed with E+Por E alone (E+O) in bilevel chambers[1]

Bremelanotide(PT-141), a cyclic heptapeptide melanocortin analogue (Palatin Technologies, Cranbury, NJ), was dissolved in saline to obtain doses of 50, 100, and 200 μg/kg/ml, and injected s.c. 5 min before each behavioral test. An equal volume of saline was administered to control animals[1].

1607799-13-2

C52H72N14O12

1085.234

bremelanotide;PT-141 Acetate

DMSO:36 mg/mL (33.17 mM)
Powder: -20°C for 3 years
In solvent: -80°C for 2 years