LE 300 是一种有效的选择性多巴胺 D1 样受体拮抗剂,在表达人多巴胺 D1 和 D5 受体的 CHO 细胞膜中,Kis 分别为 1.9 nM 和 7.5 nM。
Cas No. | 274694-98-3 |
化学名 | 7-methyl-6,7,8,9,14,15-hexahydro-5H-benzo[7,8]azecino[5,4-b]indole |
Canonical SMILES | CN1CCC2=C(CC3=CC=CC=C3CC1)NC4=CC=CC=C24 |
分子式 | C20H22N2 |
分子量 | 290.41 |
溶解度 | <14.52mg/ml in 1eq. HCl;<29.04mg/ml in DMSO |
储存条件 | Store at RT |
General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |