Telomerase-IN-2 是一种端粒酶抑制剂,通过降低角化不良蛋白的表达来抑制其活性,IC50值为 0.89?μM,具有抗癌作用。
产品描述
Telomerase-IN-2 shows potent inhibitory activity against telomerase by decreasing the expression of dyskerin (IC50: 0.89 μM).
体外活性
Telomerase-IN-2 exhibits high activity against Hela, SMMC-7721, SGC-7901, U87 and HepG2 cell lines in the anticancer activity assay in vitro[1].
Cas No.
1610878-54-0
分子式
C34H39N3O9
分子量
633.69
别名
Telomerase inhibitor 2;端粒酶抑制剂2
储存和溶解度
DMSO:235 mg/mL (370.84 mM),Need ultrasonic
Powder: -20°C for 3 years
In solvent: -80°C for 2 years