Halopemide 是一种有效的 PLD 抑制剂（对人 PLD1 和 PLD2 的 IC50 = 220 和 310 nM）。 Halopemid 是多巴胺受体的拮抗剂。Halopemid 可用于精神药物研究。

Halopemide is a potent inhibitor of PLD (IC50 = 220 and 310 nM for human PLD1 and PLD2). Halopemid is an antagonist of dopamine receptors. Halopemid can be used in psychotropic research.

In transdifferentiated MOVAS cells, Halopemide (1-2 μM; 21 days) influences calcification[1].

In the majority of monkeys tested, Halopemide (10 mg/kg; p.o.) causes dyskinesias[2].

59831-65-1

C21H22ClFN4O2

416.88

(< 1 mg/ml refers to the product slightly soluble or insoluble )
Powder: -20°C for 3 years
In solvent: -80°C for 2 years