Varespladib methyl 是 Varespladib 的生物可利用前药，是一种特异性 II 组分泌型磷脂酶 A2 抑制剂。

Varespladib methyl, a bioavailable prodrug of Varespladib, is a selective group II secretory phospholipase A2 inhibitor.

Varespladib methyl display high-level secretory PLA2 inhibition at nanomolar and picomolar concentrations against 28 medically important snake venoms from six continents [1].

172733-08-3

C22H22N2O5

394.42

LY333013;A-002

DMSO:95 mg/mL (240.58 mM),Need ultrasonic
Powder: -20°C for 3 years
In solvent: -80°C for 2 years