CARM1-IN-1 是 CARM1 的选择性抑制剂，IC50 为 8.6 μM。 CARM1-IN-1 对 PRMT1 和 SET7 的活性较弱，IC50 >600 μM。

CARM1-IN-1 is a selective inhibitor of CARM1 with IC50 of 8.6 μM. CARM1-IN-1 shows weak activity against PRMT1 and SET7 with IC50 >600 μM.

In human LNCaP cells, CARM1-IN-1 significantly reduces the PSA promoter activity in a dose-dependent manner[1].

1020399-49-8

C26H21Br2NO3

555.26

CARM1-IN-7G

DMSO:30 mg/mL (54 mM),Need ultrasonic
Powder: -20°C for 3 years
In solvent: -80°C for 2 years