| CAS NO: | 1962928-21-7 |
| 包装 | 价格(元) |
| 100mg | 电议 |
| 250mg | 电议 |
| 500mg | 电议 |
| 生物活性 | PF-CBP1 is a highly selective inhibitor of the CREB binding protein bromodomain[1]. |
| 体外研究 (In Vitro) | PF-CBP1 modulates key inflammatory genes in primary macrophages. PF-CBP1 downregulates RGS4 in neurons, a target linked to Parkinson's disease. PF-CBP1 is 139-fold selective over BRD4 in the biochemical assays and >105-fold selective by ITC. F-CBP1 is also a potent inhibitor of EP300 (a result observed for other CBP inhibitors[1]. |
| 分子量 | 488.62 |
| Formula | C29H36N4O3 |
| CAS 号 | 1962928-21-7 |
| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |
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