Metaraminol tartrate

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CAS NO:

33402-03-8

包装与价格：

包装	价格(元)
10 mM * 1 mL in DMSO	电议
100mg	电议
200mg	电议
500mg	电议
1 g	电议

产品名称

Metaradrine tartrate

产品介绍

Metaraminol tartrate (Metaradrine tartrate) 是一种 α-肾上腺素能 (α-adrenergic) 激动剂。Metaraminol tartrate 是一种直接或间接影响肾上腺素受体的拟交感神经胺，其中 α 效应占主导地位。Metaraminol tartrate 可作为血管加压剂。

生物活性

Metaraminol tartrate (Metaradrine tartrate) is anα-adrenergicagonist^[1]. Metaraminol tartrate is a sympathomimetic amine that directly and indirectly affects adrenergic receptors, with alpha effects being predominant.Metaraminol tartrate acts as a vasopressor agent^[2].

IC₅₀& Target

Adrenergic Receptor^[1]

体外研究
(In Vitro)

Stimulation of α-adrenoceptors by metaraminol, a drug with properties similar to noradrenaline, caused acceleration of cell proliferation in colonie crypts but not in tumors^[3].

体内研究
(In Vivo)

Lethal endotoxin shock is prevented in six of the 10 animals studied by the simultaneous use of Metaraminol^[2].

Animal Model:	Ten adult dogs weighing between 7.8 and 13 kg^[2]
Dosage:	Solution containing 25 mg in 250 mL of 5 percent dextrose and water
Administration:	Intravenous infusion
Result:	Lethal endotoxin shock was prevented,

分子量

317.29

性状

Solid

Formula

C₁₃H₁₉NO₈

CAS 号

33402-03-8

中文名称

重酒石酸间羟胺；酒石酸美拉明

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

4°C, sealed storage, away from moisture

*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)

溶解性数据

In Vitro:

DMSO : ≥ 28 mg/mL(88.25 mM)

*"≥" means soluble, but saturation unknown.

配制储备液

浓度溶剂体积质量

1 mg

5 mg

10 mg

1 mM	3.1517 mL	15.7585 mL	31.5169 mL
5 mM	0.6303 mL	3.1517 mL	6.3034 mL
10 mM	0.3152 mL	1.5758 mL	3.1517 mL

请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液；一旦配成溶液，请分装保存，避免反复冻融造成的产品失效。
储备液的保存方式和期限：-80℃, 6 months; -20℃, 1 month (sealed storage, away from moisture)。-80℃ 储存时，请在 6 个月内使用，-20℃ 储存时，请在 1 个月内使用。