CAS NO: | 103429-32-9 |
包装 | 价格(元) |
100mg | 电议 |
250mg | 电议 |
500mg | 电议 |
生物活性 | CTAP is a potent, highly selective, and BBB penetrantμopioid receptorantagonist, with anIC50of 3.5 nM. CTAP displays over 1200-fold selectivity overδ opioid(IC50=4500 nM) andsomatostatin receptors. CTAP can be used for the study of L-DOPA-induced dyskinesia (LID) and opiate overdose or addiction[1][2]. | ||||||||
IC50& Target |
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体内研究 (In Vivo) | CTAP (0-1 mg/kg, IP, single) blocks morphine’s antinociceptive effect[1].
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分子量 | 1104.30 | ||||||||
Formula | C51H69N13O11S2 | ||||||||
CAS 号 | 103429-32-9 | ||||||||
Sequence | {d-Phe}-Cys-Tyr-{d-Trp}-Arg-Thr-{Pen}-Thr-NH2 (Disulfide bridge:Cys2-Pen7) | ||||||||
Sequence Shortening | {d-Phe}-CY-{d-Trp}-RT-{Pen}-T-NH2 (Disulfide bridge:Cys2-Pen7) | ||||||||
运输条件 | Room temperature in continental US; may vary elsewhere. | ||||||||
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |