您好,欢迎来到试剂仪器网! [登录] [免费注册]
试剂仪器网
位置:首页 > 产品库 > Maropitant-13C,d3
立即咨询
咨询类型:
     
*姓名:
*电话:
*单位:
Email:
*留言内容:
请详细说明您的需求。
*验证码:
 
Maropitant-13C,d3
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Maropitant-13C,d3图片
包装与价格:
包装价格(元)
1mg电议
5mg电议

产品介绍
Maropitant-13C,d3 是一种 13C- 和氘代标记的 Maropitant。Maropitant 是一种选择性的具有口服活性的神经激肽 (NK1) 受体拮抗剂。Maropitant 通过阻止催吐中心与化学感受器触发区 (CRTZ) 中 P 物质的结合而起作用。Maropitant 在预防呕吐方面非常有效。
生物活性

Maropitant-13C,d3 is the 13C- and deuterium labeled Maropitant. Maropitant is a selective and orally active neurokinin (NK1) receptor antagonist. Maropitant acts by blocking the binding of substance P within the emetic center and the chemoreceptor trigger zone (CRTZ). Maropitant is highly effective in preventing vomiting[1][2].

体外研究
(In Vitro)

Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs[92].

分子量

472.68

Formula

C3113CH37D3N2O

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.