Toremifene-d6 citrate

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本产品不向个人销售，仅用作科学研究，不用于任何人体实验及非科研性质的动物实验。

CAS NO:	1246833-71-5
包装:	1mg
市场价:	5500元

产品名称

枸橼酸托瑞米芬 d6 (柠檬酸盐)

产品介绍

Toremifene-d6 (Z-Toremifene-d6) citrate 是 Toremifene citrate 的氘代物。Toremifene citrate (Z-Toremifene citrate) 是第二代选择性雌激素受体调节剂，对雌激素受体的IC₅₀为 1μM。Toremifene citrate 还可以有效抑制传染性EBOV Zaire和Marburg (MARV)，IC₅₀分别为 0.07 μM 和 2.6 μM。

生物活性	Toremifene-d6 (Z-Toremifene-d6) citrate is the deuterium labeled Toremifene citrate. Toremifene citrate (Z-Toremifene citrate) is a second-generation selectiveestrogen-receptor modulator (SERM)in development for the prevention of osteoporosis. Toremifene citrate also potent inhibits infectiousEBOV ZaireandMarburg (MARV)withIC₅₀of 0.07 μM and 2.6 μM, respectively^[1]^[2].
体外研究 (In Vitro)	Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs^[1].
分子量	604.12
Formula	C₃₂H₃₀D₆ClNO₈
CAS 号	1246833-71-5
中文名称	枸橼酸托瑞米芬 d6 (柠檬酸盐)
运输条件	Room temperature in continental US; may vary elsewhere.
储存方式	Please store the product under the recommended conditions in the Certificate of Analysis.