Imlunestrant

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Imlunestrant

本产品不向个人销售，仅用作科学研究，不用于任何人体实验及非科研性质的动物实验。

CAS NO:

2408840-26-4

包装与价格：

包装	价格(元)
100mg	电议
250mg	电议
500mg	电议

产品名称

LY-3484356

产品介绍

Imlunestrant (LY3484356) 是具有口服活性的选择性雌激素受体的降解剂(SERD)。Imlunestrant (LY3484356) 可用以ER+ 和HER2 乳腺癌。

生物活性

Imlunestrant (LY3484356) is an orally active selectiveestrogen receptor(ER)degrader (SERD). Imlunestrant (LY3484356) could be used in the study for ER+, HER2-advanced breastcancer^[1].

体外研究
(In Vitro)

Imlunestrant (LY3484356) shows favorable efficacy and pharmacokinetic (PK) properties, including antitumor activity in ESR1 mutants^[1].
Imlunestrant (LY3484356) is a potent degrader and selective pure antagonist of wild type and mutant ERα^[2].

Clinical Trial

分子量

524.51

Formula

C₂₉H₂₄F₄N₂O₃

CAS 号

2408840-26-4

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.