Thioperamide (MR-12842) 是一种有效的、可口服的、脑渗透剂和选择性 H3 受体拮抗剂，其 Ki 为 4.3 nM，用于抑制 [3H] 组胺的释放。
| Cas No. | 106243-16-7 |
| 别名 | 硫丙咪胺,MR-12842 |
| 化学名 | N-cyclohexyl-4-(1H-imidazol-5-yl)piperidine-1-carbothioamide |
| Canonical SMILES | S=C(NC1CCCCC1)N2CCC(C3=CN=CN3)CC2 |
| 分子式 | C15H24N4S |
| 分子量 | 292.44 |
| 溶解度 | <29.24mg/ml in DMSO;<29.24mg/ml in ethanol |
| 储存条件 | Store at -20°C |
| General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
| Shipping Condition | Evaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request |
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