Trimipramine-d3 maleate is the deuterium labeled Trimipramine maleate. Trimipramine maleate is a5-HT receptor antagonist, with pK_is of 6.39, 8.10, 4.66 for 5-HT_1C, 5-HT₂and 5-HT_1A, respectively^[1][2].

Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs^[1].

413.52

C₂₄H₂₇D₃N₂O₄

1185245-93-5

马来酸三甲丙咪嗪 d3 (马来酸盐)

Room temperature in continental US; may vary elsewhere.

Please store the product under the recommended conditions in the Certificate of Analysis.