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Eletriptan-d3
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Eletriptan-d3图片
CAS NO:1287040-94-1
包装与价格:
包装价格(元)
1mg电议
10mg电议

产品名称
UK-116044-d3
产品介绍
Eletriptan-d3 (UK-116044-d3) 是 Eletriptan hydrobromide 的氘代物。Eletriptan hydrobromide 是一种选择性的 5-HT1B 和 5-HT1D 受体激动剂,Ki分别为 0.92 nM 和 3.14 nM。
生物活性

Eletriptan-d3 (UK-116044-d3) is the deuterium labeled Eletriptan hydrobromide. Eletriptan hydrobromide is a selective 5-HT1B and 5-HT1D receptor agonist with Kiof 0.92 nM and 3.14 nM, respectively[1][2].

体外研究
(In Vitro)

Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs[1].

分子量

385.54

Formula

C22H23D3N2O2S

CAS 号

1287040-94-1

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.