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Tegaserod-13C,d3 maleate
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Tegaserod-13C,d3 maleate图片
包装与价格:
包装价格(元)
1mg电议
5mg电议

产品名称
SDZ-HTF-919-13C,d3
HTF-919-13C,d3
产品介绍
Tegaserod-13C,d3 (maleate) 是一种 13C- 和氘代标记的 Tegaserod (maleate)。Tegaserod maleate 是选择性的、5-HT4受体的部分激动剂和5-HT2B受体的拮抗剂。Tegaserod maleate 在胃肠道中表现出促进的作用。
生物活性

Tegaserod-13C,d3 (maleate) is the 13C- and deuterium labeled Tegaserod (maleate). Tegaserod maleate is a selective 5-HT4 receptor partial agonist and a 5-HT2B receptor antagonist. Tegaserod maleate exhibits a promotile effect throughout the gastrointestinal (GI) tract[1][2][5].

体外研究
(In Vitro)

Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs[50].

分子量

421.47

Formula

C1913CH24D3N5O5

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.