PNU 142633 是一种高亲和力、选择性和口服活性的 5-HT1D 受体激动剂,对人 5-HT1D 受体和人 5-HT1B 受体的 Kis 分别为 6 nM 和 \u003e 18 000 nM。
Cas No. | 187665-65-2 |
化学名 | (S)-1-(2-(4-(4-carbamoylphenyl)piperazin-1-yl)ethyl)-N-methylisochroman-6-carboxamide |
Canonical SMILES | O=C(C1=CC2=C(C=C1)[C@H](CCN3CCN(C4=CC=C(C(N)=O)C=C4)CC3)OCC2)NC |
分子式 | C24H30N4O3 |
分子量 | 422.53 |
溶解度 | <42.25mg/ml in DMSO |
储存条件 | Store at -20℃ |
General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |