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Pindolol-d7
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Pindolol-d7图片
CAS NO:1185031-19-9
包装与价格:
包装价格(元)
2.5mg电议
1mg电议
5mg电议
10mg电议
25mg电议

产品名称
吲哚洛尔 d7
产品介绍
Pindolol-d7 是 Pindolol 的氘代物。Pindolol (LB-46) 是一种非选择性β-阻断剂, 局部的β-肾上腺素能受体激动剂活性, 也作为5-HT1A受体部分拮抗剂 (Ki=33nM)。
生物活性

Pindolol-d7 (LB-46-d7) is the deuterium labeled Pindolol. Pindolol (LB-46) is a nonselective β-blocker with partial beta-adrenergic receptor agonist activity, also functions as a 5-HT1A receptor weak partial antagonist (Ki=33 nM)[1][2].

体外研究
(In Vitro)

Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs[1].

分子量

255.36

Formula

C14H13D7N2O2

CAS 号

1185031-19-9

中文名称

吲哚洛尔 d7

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.