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Fosphenytoin-d10 disodium
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Fosphenytoin-d10 disodium图片
包装与价格:
包装价格(元)
1mg电议
5mg电议

产品介绍
Fosphenytoin-d10 (disodium) 是 Fosphenytoin (disodium) 氘代物。Fosphenytoin sodium 是 phenytoin 的前提药物,具有抗惊厥等功效。其主要机制是阻断神经元钠通道,从而限制动作电位的重复放电。
生物活性

Fosphenytoin-d10 (disodium) is deuterium labeled Fosphenytoin (disodium). Fosphenytoin sodium is a phenytoin prodrug with similar anticonvulsant properties. Its main mechanism is to block frequency-dependent, use-dependent and voltage-dependent neuronal sodium channels, and therefore limit repetitive firing of action potentials.

体外研究
(In Vitro)

Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs[1].

分子量

416.30

Formula

C16H3D10N2Na2O6P

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.