Tolvaptan-D7 (OPC-41061-D7) is the deuterium labeled Tolvaptan. Tolvaptan is a selective, competitive argininevasopressin receptor2 antagonist with an IC₅₀of 1.28μM for the inhibition of AVP-induced platelet aggregation^[1][2].

Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs^[1].

455.98

C₂₆H₁₈D₇ClN₂O₃

1246818-18-7

托伐普坦 D7

Room temperature in continental US; may vary elsewhere.

Please store the product under the recommended conditions in the Certificate of Analysis.