Antagonist G is a potentvasopressinantagonist. Antagonist G is also a weak antagonist of GRP and Bradykinin. Antagonist G inducesAP-1transcription and sensitizes cells to chemotherapy^[1][2].

Antagonist G (0-100 μM) induces apoptosis is redox-sensitive and caspase-dependently in SCLC cells^[2].
Antagonist G activates JNK1 in SCLC cells^[2].
Antagonist G is not intrinsically a free radical oxygen donor but stimulates free radical generation specifically within SCLC cells (6.2-fold) and increases the activity of the redox-sensitive transcription factor AP-1 by 61%^[2].

951.19

Solid

C₄₉H₆₆N₁₂O₆S

115150-59-9

RW-{Me-Phe}-WLM-NH2

Room temperature in continental US; may vary elsewhere.

Sealed storage, away from moisture and light

*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light)

H₂O : 50 mg/mL(52.57 mM;Need ultrasonic)

请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液；一旦配成溶液，请分装保存，避免反复冻融造成的产品失效。
储备液的保存方式和期限：-80℃, 6 months; -20℃, 1 month (sealed storage, away from moisture and light)。-80℃ 储存时，请在 6 个月内使用，-20℃ 储存时，请在 1 个月内使用。