CAS NO: | 1160271-30-6 |
包装: | 1mg |
生物活性 | PPTN is a potent, high-affinity, competitive and highly selectiveP2Y14 receptorantagonist with aKBvalue of 434 pM. PPTN exhibits no agonist or antagonist effect at the P2Y1, P2Y2, P2Y4, P2Y6, P2Y11, P2Y12, or P2Y13 receptors. Anti-inflammatory and immune activity[1]. |
IC50& Target | KB: 434 pM (P2Y14 receptor)[1] |
体外研究 (In Vitro) | PPTN exhibits strong selectivity for the P2Y14-R over the other seven nucleotide-activated P2Y receptors. 1 μM PPTN exhibits no agonist or antagonist effect at the P2Y1, P2Y2, P2Y4, P2Y6, P2Y11, P2Y12, or P2Y13 receptors[1]. |
分子量 | 475.50 |
Formula | C29H24F3NO2 |
CAS 号 | 1160271-30-6 |
运输条件 | Room temperature in continental US; may vary elsewhere. |
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |