| CAS NO: | 479080-38-1 |
| 包装 | 价格(元) |
| 100mg | 电议 |
| 250mg | 电议 |
| 500mg | 电议 |
| 生物活性 | OT antagonist 1 (Compound 4) is a potent, selectiveOxytocinantagonist with aKiof 50 nM. |
| IC50& Target | Ki: 50 nM (Oxytocin)[1] |
| 体外研究 (In Vitro) | Oxytocin (OT) is a nonapeptide hormone that acts on the OT receptor, a seven-transmembrane (7TM) (Gq-coupled) receptor. The OT receptor has no subtypes but is related to the vasopressin receptors V1A, V1Band V2. OT antagonists have therapeutic potential in a number of areas including pre-term labour: Benign Prostatic Hyperplasia and sexual dysfunction. As a result there is significant interest in the identification of potent, selective, orally bioavailable OT antagonists[1]. |
| 分子量 | 390.44 |
| Formula | C22H22N4O3 |
| CAS 号 | 479080-38-1 |
| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |
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