CAS NO: | 950492-85-0 |
包装 | 价格(元) |
10 mM * 1 mL in Water | 电议 |
1mg | 电议 |
5mg | 电议 |
10mg | 电议 |
25mg | 电议 |
50mg | 电议 |
100mg | 电议 |
生物活性 | DAMGO TFA is aμ-opioid receptor(μ-OPR) selective agonist with aKdof 3.46 nM for native μ-OPR[1]. | ||||||||||||||||
体外研究 (In Vitro) | DAMGO (1-10 μM) TFA significantly reduces the activation of neuronal Akt and ERK1/2 by CXCL12 and inhibits CXCL12-promoted neuronal survival, but does not down-regulate CXCR4 protein expression[2]. | ||||||||||||||||
体内研究 (In Vivo) | DAMGO (i.v., 0.5-2 mg/kg) TFA can produce significant anti-injury effects on injured paws of male Sprague-Dawley rats weighing 200-225 g in a dose-dependent manner, producing an effective and long-lasting analgesic effect[4]. | ||||||||||||||||
分子量 | 627.61 | ||||||||||||||||
性状 | Solid | ||||||||||||||||
Formula | C28H36F3N5O8 | ||||||||||||||||
CAS 号 | 950492-85-0 | ||||||||||||||||
Sequence | Tyr-{d-Ala}-Gly-{Me-Phe}-Gly-ol | ||||||||||||||||
Sequence Shortening | Y-{d-Ala}-G-{Me-Phe}-G-ol | ||||||||||||||||
运输条件 | Room temperature in continental US; may vary elsewhere. | ||||||||||||||||
储存方式 | Sealed storage, away from moisture
*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture) | ||||||||||||||||
溶解性数据 | In Vitro: H2O : 125 mg/mL(199.17 mM;Need ultrasonic) 配制储备液
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以下溶剂前显示的百
*以上所有助溶剂都可在本网站选购。 |