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BAY 1214784
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
BAY 1214784图片
CAS NO:1631164-25-4
包装与价格:
包装价格(元)
100mg电议
250mg电议
500mg电议

产品介绍
BAY 1214784 是人促性腺激素释放激素受体 (hGnRH-R) 的有效、选择性和口服活性拮抗剂。BAY 1214784 是螺二氢吲哚衍生物化合物。BAY 1214784 可有效降低血浆促黄体激素水平高达 49%,同时具有较低的药代动力学变异性和良好的耐受性。BAY 1214784 具有研究子宫肌瘤的潜力。
生物活性

BAY 1214784 is a potent, selective, and orally active antagonist of the human gonadotropin-releasing hormone receptor (hGnRH-R). BAY 1214784 is a spiroindoline derivative compound. BAY 1214784 effectively lowers plasma luteinizing hormone levels by up to 49%, at the same time being associated with low pharmacokinetic variability and good tolerability. BAY 1214784 has the potential for the research of uterine fibroids[1].

分子量

672.11

Formula

C29H26ClF4N3O5S2

CAS 号

1631164-25-4

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.