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Elagolix-13C,d3 sodium
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Elagolix-13C,d3 sodium图片
包装与价格:
包装价格(元)
1mg电议
5mg电议

产品名称
NBI-56418-13C,d3 sodium
产品介绍
Elagolix-13C,d3 (sodium) 是一种 13C- 和氘代标记的 Elagolix sodium。Elagolix sodium 是一种人的GnRH受体 (GnRHR) 拮抗剂,其IC50Ki值分别为 0.25 和 3.7 nM。
生物活性

Elagolix-13C,d3 (sodium) is the 13C- and deuterium labeled Elagolix sodium. Elagolix sodium is a humanGnRH receptor(GnRHR) antagonist with an IC50 and Ki of 0.25 and 3.7 nM, respectively.

体外研究
(In Vitro)

Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs[56].

分子量

657.58

Formula

C3113CH26D3F5N3NaO5

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.