CAS NO: | 158848-32-9 |
包装 | 价格(元) |
10mg | 电议 |
50mg | 电议 |
Cas No. | 158848-32-9 |
别名 | ({1-[2-(5-氟-1H-吲哚-3-基)乙基]-4-甲氧基-4-哌啶基}甲基)(苯基)锍醇 |
化学名 | 5-fluoro-3-(2-(4-methoxy-4-((phenylsulfinyl)methyl)piperidin-1-yl)ethyl)-1H-indole |
Canonical SMILES | FC1=CC=C2NC=C(C2=C1)CCN3CCC(CC3)(CS(C4=CC=CC=C4)=O)OC |
分子式 | C23H27FN2O2S |
分子量 | 414.54 |
溶解度 | 30mg/ml in DMSO |
储存条件 | Desiccate at -20°C |
General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |
产品描述 | GR 159897 is a highly potent, selective, competitive, brain-penetrated non-peptide antagonist at tachykinin NK2 receptors, inhibits binding of [3H]GR100679 to hNK2-CHO cells and rat colon membranes with pKis of 9.51 and 10, respectively. Antagonizes bronchoconstriction, with anxiolytic-like activity[1]. References: |