CP 316819 是一种有效的糖原磷酸化酶 (GPase) 抑制剂,具有抗高血糖作用(对人骨骼肌糖原磷酸化酶 (huSMGPa) 和肝糖原磷酸化酶 (huLGPa) 的 IC50 值分别为 17 和 34 nM)。
Cas No. | 186392-43-8 |
别名 | GPi 819 |
化学名 | 5-chloro-N-((2S,3S)-3-hydroxy-4-((methoxymethyl)amino)-4-oxo-1-phenylbutan-2-yl)-1H-indole-2-carboxamide |
Canonical SMILES | ClC1=CC=C2NC(C(N[C@H]([C@@H](C(NCOC)=O)O)CC3=CC=CC=C3)=O)=CC2=C1 |
分子式 | C21H22ClN3O4 |
分子量 | 415.87 |
溶解度 | <41.59mg/ml in DMSO;<41.59mg/ml in ethanol |
储存条件 | Store at RT |
General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |